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Mariangela Ceruso Selected Research

carbonic anhydrase XII

6/2015New series of sulfonamides containing amino acid moiety act as effective and selective inhibitors of tumor-associated carbonic anhydrase XII.
4/2014Arylamino bisphosphonates: potent and selective inhibitors of the tumor-associated carbonic anhydrase XII.
3/2014Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII.
12/2013Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII--a new scaffold for designing isoform-selective inhibitors.

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Mariangela Ceruso Research Topics

Disease

40Neoplasms (Cancer)
04/2020 - 12/2013
5Glaucoma
01/2018 - 01/2016
4Breast Neoplasms (Breast Cancer)
01/2018 - 05/2014
2Pathologic Processes
12/2015 - 04/2014
1Cholera
12/2017
1Carcinogenesis
03/2016
1Arthritis (Polyarthritis)
01/2016
1Acidosis
01/2016
1Pain (Aches)
01/2016
1Epilepsy (Aura)
01/2016
1Communicable Diseases (Infectious Diseases)
08/2014
1Bone Resorption
06/2014
1Neoplasm Metastasis (Metastasis)
06/2014

Drug/Important Bio-Agent (IBA)

39Protein Isoforms (Isoforms)IBA
08/2019 - 12/2013
31Carbonic Anhydrases (Carbonic Anhydrase)IBA
04/2020 - 03/2014
19SulfonamidesIBA
04/2020 - 05/2014
10EnzymesIBA
01/2018 - 06/2014
9IsoenzymesIBA
08/2019 - 06/2014
7Pharmaceutical PreparationsIBA
01/2018 - 07/2014
5BenzenesulfonamidesIBA
01/2018 - 12/2014
4Biological ProductsIBA
08/2019 - 07/2015
4Carbonic Anhydrase IXIBA
01/2018 - 01/2016
4carbonic anhydrase XIIIBA
06/2015 - 12/2013
3Acetazolamide (Diamox)FDA LinkGeneric
01/2016 - 11/2014
3Antineoplastic Agents (Antineoplastics)IBA
01/2016 - 06/2015
2SaccharinIBA
12/2017 - 03/2014
2ThymidineIBA
07/2015 - 05/2014
2DNA (Deoxyribonucleic Acid)IBA
07/2015 - 05/2014
2Diphosphonates (Bisphosphonates)IBA
06/2014 - 04/2014
1Carbonic Anhydrase InhibitorsIBA
08/2019
1OxidesIBA
08/2019
1SLC-0111IBA
01/2018
1dorzolamide (Trusopt)FDA LinkGeneric
01/2018
1Ophthalmic Solutions (Eye Drops)IBA
01/2018
1Adrenergic Receptors (Adrenergic Receptor)IBA
01/2018
1Timolol (Blocadren)FDA LinkGeneric
01/2018
1Adrenergic Agents (Adrenergic Drugs)IBA
01/2018
1Sodium Bicarbonate (Baking Soda)FDA LinkGeneric
12/2017
1IsatinIBA
03/2016
1imidazoleIBA
01/2016
1ChloridesIBA
01/2016
1trimellitic anhydrideIBA
01/2016
1coumarinIBA
01/2016
1gamma-Aminobutyric Acid (GABA)IBA
01/2016
1ortho-AminobenzoatesIBA
01/2016
1AminesIBA
01/2016
1IminesIBA
12/2015
1CoumarinsIBA
11/2015
1Phenol (Carbolic Acid)FDA Link
09/2015
1Amino AcidsFDA Link
06/2015
1ChromonesIBA
01/2015
1Carboxylic AcidsIBA
12/2014
1AldehydesIBA
12/2014
1SulfanilamideFDA Link
12/2014
1Heterocyclic Compounds (Compounds, Heterocyclic)IBA
12/2014
1pyrazoleIBA
12/2014
1NitrilesIBA
12/2014
1OximesIBA
12/2014
1carboxyl radical (COO-)IBA
11/2014
1Schiff Bases (Schiff Base)IBA
11/2014
1sulfamic acid (ammonium sulfamate)IBA
09/2014
1Doxorubicin (Adriamycin)FDA LinkGeneric
07/2014
1Matrix Metalloproteinases (MMPs)IBA
06/2014
1Matrix Metalloproteinase InhibitorsIBA
06/2014
1Enzyme Inhibitors (Inhibitors, Enzyme)IBA
06/2014
1AcidsIBA
06/2014
1CollagenIBA
05/2014
1aniline (aniline hydrobromide)IBA
05/2014
1TriazinesIBA
05/2014
1Sildenafil Citrate (Viagra)FDA Link
05/2014
1ZincIBA
03/2014
1disalicylaldehyde ethylenediamine (salen)IBA
12/2013

Therapy/Procedure

1Investigational Therapies (Experimental Therapy)
01/2016